Samfur Description
1. Fasoracetam Foda Bidiyo-AASraw
2. Raw Fasoracetam Foda Basic Characters
name: | Fasoracetam foda |
CAS: | 110958-19-5 |
Formula kwayoyin: | C14H27N3O2 |
Kwayoyin Weight: | 158.15 |
Shawarwar Melt: | 160-166 ° C |
Ajiye Temp: | Store a dakin da zazzabi ko mai sanyaya |
Color: | White ko kashe-farin foda |
Abin da is Fasoracetam foda?
Fasoracetam wani nau'in nootropic na roba ne na racetams. Wani kamfanin harhada magunguna na kasar Japan da farko ya samar da shi don magance cutar dementia, amma rashin inganci ya hana ci gabansa.
Duk da haka, kwanan nan ya sake bayyana a cikin gwaje-gwajen asibiti, tare da bincike yana duba yiwuwar magance cututtuka daban-daban da kuma inganta fahimtar gaba ɗaya.
Aevi Genomic Medicine ne ya ɗauki matakin wanda ya fara gwaji na asibiti don bincika yadda wannan magani zai iya shafar mutane akan cutar ta Autism, waɗanda ke da matsalar rashin hankali (ADHD), da damuwa.
Ta yaya Fasoracetam yake aiki a cikin kwakwalwa?
Fasoracetam yana aiki ta hanyar hulɗar da daidaita tsarin tsarin neurochemical guda uku: tsarin glutamatergic, cholinergic, da gabaergic.
Dukkanin ukun suna iya aiki a cikin ƙarfin haɓakar fahimi tare da fa'idodi masu yuwuwa kamar haɓaka aikin fahimi, rage hazo na kwakwalwa, da haɓakar tsabtar tunani.
Kamar sauran abubuwan nootropic, fasoracetam yana ƙara matakan acetylcholine. Wannan aikin cholinergic yana taimakawa haɓaka fahimta, ƙwaƙwalwa, mayar da hankali, yanayi, faɗakarwa, neuroplasticity, da ƙwaƙwalwar ajiyar lokaci mai tsawo.
A lokaci guda kuma, yana hana raguwar acetylcholine ta hanyar cholinesterase, yana ƙarfafa ɗaukarsa ta hanyar masu karɓa na cholinergic.
Sauran neurotransmitter da yake aiki akan shine gamma-aminobutyric acid (GABA) ta hanyar haɓaka masu karɓar GABA (B).
Masu karɓar GABA suna nan a ko'ina cikin tsarin juyayi na tsakiya kuma, lokacin da aka kunna su, suna haifar da ƙuntatawa mai yawa a cikin tsarin kulawa na tsakiya.
A wasu kalmomi, GABA yana kwantar da ƙwayoyin neurons don inganta jin dadi da jin dadi. Bugu da ƙari, waɗannan hanyoyin suna taimakawa GABA don shawo kan damuwa, tsoro, rashin barci, da damuwa.
Hanya na uku ya ƙunshi tsarin glutamate. Fasoracetam kuma yana daidaita masu karɓar glutamate na farko na metabotropic, yana shafar ayyukan fahimi, neuroprotection, filastik synaptic, da damuwa gabaɗaya.
Rashin daidaituwa na rashin daidaituwa na neurotransmitter glutamate ana iya danganta shi da rikice-rikice na tunani da na jiki da yawa, gami da damuwa, ADHD, farfadiya, da cutar Alzheimer, don suna kaɗan.
The Amfanin Fasoracetam
Ƙila inganta ingantaccen ƙwaƙwalwar ajiya da kuma Janar ƙusarwa
A cikin gwajin dabba, fasoracetam ya hana ko rage amnesia da mantuwa
Ko da yake babu bayanan da aka samu a bainar jama'a game da irin wannan gwaje-gwajen akan batutuwan ɗan adam, yawancin masu amfani sun ce sun sami ingantaccen ƙwaƙwalwar ajiya lokacin ɗaukar ta.
Kamar sauran racetam nootropics, fasoracetam yana ƙara yawan adadin acetylcholine, neurotransmitter mafi alhakin ƙwaƙwalwar ajiya, koyo, da fahimta.
Yarda Cigaba da damuwa da damuwa
Fasoracetam na iya inganta yanayi, rage damuwa, da kuma ɗaga bakin ciki ta hanyar yin aiki akan biyu daga cikin sinadarai masu tasiri mafi ƙarfi na kwakwalwa, glutamate da gamma-aminobutyric acid (GABA).
Ta hanyar daidaitawa lokaci guda GABA, wanda shine mai hanawa neurotransmitter, da kuma hana wuce haddi na samar da excitatory neurotransmitter glutamate, fasoracetam yana ba da abin da masu amfani suka kwatanta a matsayin santsi, rashin jin dadi na inganta yanayi, shakatawa, da kwanciyar hankali.
Babu wani bincike na jama'a game da tasirin fasoracetam akan yanayi, damuwa, ko damuwa a cikin mutane, amma yawancin masu amfani suna ba da rahoton cewa suna jin dadi, rashin damuwa, da rashin damuwa lokacin shan shi.
M ADHD jiyya
Ɗaya daga cikin ƙananan binciken ɗan adam da ake samuwa a kan fasoracetam ya nuna cewa yana iya zama yiwuwar magani ga ADHD
Binciken, wanda ya shafi batutuwa na 30 tsakanin shekarun 12 da 17, sun gwada tasirin fasoracetam a cikin magance ADHD tsakanin matasa waɗanda suka nuna takamaiman maye gurbi a cikin hanyar sadarwar glutamatergic. Wannan maye gurbin yana da alaƙa mai ƙarfi da ADHD kuma yana nan a cikin ɗimbin kashi na matasa masu fama da cutar.
Abubuwan da suka dauki fasoracetam a cikin makonni biyar na binciken sun nuna ingantaccen ci gaba a duk matakan asibiti yayin gwaji. Rage alamun ADHD ya ci gaba a gwajin gwaji, kuma babu wani daga cikin mahalarta binciken da ya nuna ci gaban ko dai haƙuri ko dogara.
Fasoracetam amfani dashi don inganta aikin fahimi
An gano Fasoracetam ba shi da tasiri don magance matsalolin ƙwaƙwalwar ƙwayar cuta wanda ya haifar da yanayi irin su lalata ko cutar Alzheimer. Gabaɗaya, fasoracetam yana da alama ba shi da tasiri don rage raguwar fahimi da ke da alaƙa da shekaru da kuma inganta kowane nau'in rashin lafiyar da ke da alaƙa da jijiyoyin jini.
Wannan ya ce, nazarin dabba yana nuna cewa fasoracetam zai iya zama tasiri don inganta aikin ƙwaƙwalwar ajiya. A cikin binciken da aka riga aka ambata - duba tunani [1] - masu bincike sun gano cewa gwamnatin fasoracetam ta iya juyar da raunin ƙwaƙwalwar ajiya wanda GABA agonists mai karɓa ya haifar. An gudanar da wannan binciken akan rodents, amma wannan tsarin yana wanzu a cikin mutane; yana da ma'ana cewa rage ayyukan mai karɓa na GABA (ko juya masu karɓan GABA agnoists) zai inganta aikin ƙwaƙwalwar ajiya.
Inda zan siya Fasoracetam Foda?
Binciken mu ya nuna cewa fasoracetam yana nuna babban alkawuran da za a yi don kula da cututtuka na jijiyoyi irin su ADHD bayyanar cututtuka, cututtuka na autism, da damuwa.
Hakanan yana ba da fa'idodi don haɓaka fannoni daban-daban na fahimi gabaɗaya, kamar haɓaka mayar da hankali da maida hankali, rage ɓarkewar ƙwaƙwalwa, da haɓaka ƙwaƙwalwar ajiya, duk ba tare da haɗarin juriya ko dogaro ba. Wannan ya taƙaita duk abin da ingancin nootropics alkawari don haɓaka aikin kwakwalwa.
Raw Fasoracetam foda Rahoton Gwajin-HNMR
Menene HNMR kuma Menene Bakan HNMR ke gaya muku?H Nuclear Magnetic Resonance (NMR) spectroscopy dabara ce ta nazarin sinadarai da ake amfani da ita wajen sarrafa inganci da bincike don tantance abun ciki da tsarkin samfurin da kuma tsarinsa na kwayoyin halitta. Misali, NMR na iya tantance gaurayawan da ke dauke da sanannun mahadi. Don mahaɗan da ba a san su ba, NMR ana iya amfani da su ko dai don daidaitawa da ɗakunan karatu na bakan gizo ko don fahimtar ainihin tsarin kai tsaye. Da zarar an san ainihin tsarin, ana iya amfani da NMR don ƙayyade daidaituwar kwayoyin halitta a cikin bayani tare da nazarin kaddarorin jiki a matakin kwayoyin halitta kamar musanya mai daidaituwa, canje-canjen lokaci, solubility, da yadawa.
Fasoracetam (110958-19-5) - COA
Fasoracetam (110958-19-5) - COA
Yadda za a saya Fasoracetam Foda daga AASraw?
❶Don tuntuɓar mu ta tsarin binciken imel ɗin mu, ko kuma ku bar mana lambar ku ta whatsapp, wakilin sabis na abokin ciniki (CSR) zai tuntuɓar ku cikin awanni 12.
❷Don samar mana da adadin ku da adireshin ku.
❸CSR ɗin mu zai ba ku fa'ida, lokacin biyan kuɗi, lambar bin diddigi, hanyoyin bayarwa da ƙididdigar ranar isowa (ETA).
❹An gama biyan kuɗi kuma za a aika da kayan a cikin awanni 12.
❺Kayan da aka karɓa kuma a ba da sharhi.
reference
[1] "Fasoracetam a cikin samari tare da ADHD da bambance-bambancen hanyoyin sadarwa na glutamatergic suna rushe siginar mGluR neurotransmitter". Binciken Gate. An dawo da 2020-10-16.
[2]Malykh, AG; Sadaie, MR (12 Fabrairu 2010). "Piracetam da piracetam-kamar kwayoyi: daga kimiyya na asali zuwa aikace-aikacen asibiti na zamani zuwa cututtuka na CNS". Magunguna. 70 (3): 287-312.
[3] Tardner, P. "Fasoracetam a matsayin magani ga ADHD: nazari na yau da kullum na bayanan asibiti da ake samuwa • Jarida ta Duniya na Kimiyyar Muhalli & Fasaha. An dawo da 2020-10-16.
[4] "Sakin Latsawa: Medgenics, Inc. Ya Sanar da Canjin Suna zuwa Aevi Genomic Medicine, Inc". Aevi ta hanyar MarketWired. 16 Disamba 2016.
[5]Moskowitz, DH (2017). Nemo Dalilin Halitta da Magunguna don ADHD, Autism da 22q. BookBaby (aka buga). ISBN 9781483590981.